1st Drug List

1
1st Drug List
2
acebutolol
3
ß1 antagonist with intrinsic sympathomimetic
activity (partial agonist)
4
albuterol
5
B2 agonist
6
amphetamine
7
Indirect sympathomimetic agent
8
atenolol
9
ß1 agonist
10
atropine
11
M antagonist
12
bethanechol
13
M agonist
14
Black widow spider venom
15
Stimulates exocytosis of Ach at cholinergic nerve
terminals
16
Botulinum toxin
17
Inhibits exocytosis of Ach at cholinergic nerve
terminals
18
carbachol
19
M agonist w/ some N agonist activity (not
clinically used as such)
20
clonidine
21
a2 agonist
22
Clorgyline
23
MAO-A inhibitor
24
cocaine
25
Uptake-1 inhibitor
26
decamethonium
27
Depolarizing NM blocking agent
28
dobutamine
29
B1 agonist
30
donepezil
31
Non-covalent AntiChE (long lasting)
32
echothiophate
33
Phosphorylating AntiChE
34
edrophonium
35
Non-covalent AntiChE (short-acting)
36
ephedrine
37
Indirect sympathomimetic agent also a weak a
and B agonist
38
galantamine
39
Non-covalent AntiChE (long-acting)
40
hemicholinum
41
Na/Ch cotransporter inhibitor
42
hexamethonium
43
Non-competitive ganglionic blocking agent (NN
antagonist)
44
homatropine
45
M antagonist
46
imipramine
47
Tricyclic antidepressant inhibits uptake-1
48
ipratropium
49
M antagonist (quaternary amine)
50
Isofluorophate (DFP)
51
Phosphorylating AntiChE
52
isoproterenol
53
B agonist
54
malathion
55
Phosphorylating AntiChE (insecticide)
56
mecamylamine
57
Non-competitive ganglionic blocking agent (NN
antagonist)
58
metaproterenol
59
B2 agonist
60
methacholine
61
M agonist
62
methamphetamine
63
Indirect sympathomimetic agent, increased CNS
effect over amphetamine
64
methoxamine
65
a1 agonist
66
a-methyl p-tyrosine
67
Tyrosine hydroxylase inhibitor
68
a-methyl dopa
69
Converted to a-methylNE in adrenergic nerve
terminals
70
a-methylNE
71
a2 agonist (also functions as a false NT)
72
metoprolol
73
B1 antagonist
74
moclobemide
75
MAO-A inhibitor (reversible)
76
nadolol
77
ß antagonist
78
neostigmine
79
Carbamoylating AntiChE (N)
80
parathion
81
Phosphorylating AntiChE
82
pargyline
83
MAO inhibitor
84
phenoxybenzamine
85
a antagonist (irreversible)
86
phentolamine
87
a antagonist
88
phenylephrine
89
a1 agonist
90
physostigmine
91
carbamoylation AntiChE
92
pilocarpine
93
M agonist
94
pindolol
95
ß antagonist with intrinsic sympathomimetic
activity (partial agonist)
96
pirenzepine
97
M1 antagonist
98
pralidoxime (2-PAM)
99
AChE reactivating agent
100
prazosin
101
a1 antagonist
102
propranolol
103
B antagonist
104
pseudoephedrine
105
indirect sympathomimetic agent weak a and B
agonist
106
pyridostigmine
107
Carbamoylating AntiChE agent (N)
108
reserpine
109
inhibits VMAT in adrenergic nerve terminal
110
rivastigmine
111
Carbamoylating AntiChE agent
112
scopolamine
113
M antagonist
114
selegiline
115
MAO-B inhibitor
116
succinylcholine
117
depolarizing NM blocking agent
118
tamsulosin
119
a1 antagonist
120
terbutaline
121
B2 agonist
122
timolol
123
B antagonist
124
tiotropium
125
M antagonist (quaternary amine)
126
tolterodine
127
M antagonist w/ functional selectivity for M2/M3
receptors in bladder
128
14
tranylcypromine
129
14
MAO inhibitor
130
14
tricyclic antidepressants
131
14
uptake-1 inhibitors
132
14
trimethaphan
133
14
competitive ganglionic blocking agent (NN
antagonist)
134
14
d-tubocurarine
135
14
competitive NM blocking agent
136
14
tyramine
137
14
indirect sympathomimetic agent (not a drug found
in food)
138
14
vesamicol
139
14
Inhibits VAchT in cholinergic nerve terminals
140
14
yohimbine
141
14
a2 antagonist